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RAD140 Inhibitor 6 years 29 weeks ago

Product NameRAD140
Catalog Number1182367-47-0

RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM).IC50 value: 7 nM (Ki, fot androgen receptor).Target: androgen receptor
Molecular Weight393.83
Molecular FormulaC20H16ClN5O2
QuantityGrams-Kilos

lamotrigine inhibitor 6 years 7 weeks ago

Lamotrigine is an anticonvulsant, inhibiting glutamate release, possibly through inhibition of Na+, K+ and Ca2+ currents.
Molecular Weight 256.09
Molecular Formula C9H7Cl2N5
Target Sodium Channel
Reference-Concentrations of lamotrigine in a mother on lamotrigine treatment and her newborn child

Loratadine Inhibitor 6 years 7 weeks ago

Loratadine is a histamine H1 receptor antagonist, used to treat allergies. Also acts as a selective inhibitor of B(0)AT2 with IC50 of 4 μM.
Reference Reading
1.Effects of Prednisolone on the Pharmacokinetics of Loratadine after Oral and Intravenous Administration of Loratadine in Rats
2.Physicochemical characterization and dissolution enhancement of loratadine by solid dispersion technique

Quizartinib inhibitor 6 years 25 weeks ago

Quizartinib is an orally available small molecule with potential antineoplastic activity. Class III receptor tyrosine kinase inhibitor AC220 selectively inhibits class III receptor tyrosine kinases, including FMS-related tyrosine kinase 3 (FLT3/STK1), colony-stimulating factor 1 receptor (CSF1R/FMS), stem cell factor receptor (SCFR/KIT), and platelet derived growth factor receptors (PDGFRs), resulting in inhibition of ligand-independent leukemic cell proliferation and apoptosis.

GW3965 inhibitor 6 years 25 weeks ago

GW3965 is a potent, selective LXR agonist for hLXRα and hLXRβ. When screened against a panel of nuclear receptors, it cross-reacted with only the pregnane X receptor (PXR). In Vitro: Recruit the steroid receptor coactivator 1 to human LXRα with EC50 of 125 nM in a cell-free ligand-sensing assay

Distamycin A hydrochloride 6 years 31 weeks ago

CAS Numbe r6576-51-8
Molecular Weight 518.04
Molecular Formula C22H28ClN9O4
Quantity Milligrams-Grams
Quality Standard Enterprise Standard
BOC Sciences provides Distamycin A hydrochloride at any quantity levels.

Pitavastatin inhibitor 6 years 29 weeks ago

Catalog Number147526-32-7
SynonymsNK-104 Calcium
CAS Number147526-32-7
DescriptionPitavastatin calcium is a novel member of the medication class of statins.
Molecular Weight880.98
Molecular FormulaC50H46CaF2N2O8
COAInquire
Targetcholesterol esters